Rimegepant
Rimegepant ke inhibitor e nyane ea molek'hule eacalcitoninpeptide e amanang le liphatsa tsa lefutso (CGRP) receptor e thibelang ketso ea CGRP, vasodilator e matla eo ho lumeloang hore e na le karolo ea hlooho ea hlooho ea migraine. Rimegepant e amoheloa bakeng sa kalafo ea tlhaselo e matla ea migraine. Litekong tsa bongaka, rimegepant e ne e mamelloa hantle ka maemo a sa tloaelehang feela a maemo a phahameng a serum aminotransferase nakong ea kalafo mme ho se na liketsahalo tse tlalehiloeng tsa kotsi ea sebete e hlakileng.
Rimegepant ke mohanyetsi oa molomo oa receptor ea CGRP e entsoeng ke Biohaven Pharmaceuticals. E amohetse tumello ea FDA ka la 27 Hlakubele 2020 bakeng sa kalafo e bohloko ea hlooho ea migraine. Le hoja bahanyetsi ba 'maloa ba batsoali ba CGRP le receptor ea eona ba amoheletsoe bakeng sa phekolo ea migraine (mohlala [erenumab], [fremanezumab], [galcanezumab]), rimegepant le [ubrogepant] ke bona feela litho tsa lelapa la "gepants" la meriana e setseng nts'etsopele, le bahanyetsi feela ba CGRP ba nang le bioavailability ea molomo. Tekanyetso ea hajoale ea kalafo ea migraine e kenyelletsa kalafo ea ho ntša mpa ka "triptans", joalo ka [sumatriptan], empa meriana ena e hanyetsanoa ho bakuli ba nang le lefu la cerebrovascular le pelo le methapo ea pelo ka lebaka la thepa ea bona ea vasoconstrictive. Khahlano ea tsela ea CGRP e fetohile sepheo se khahlehang bakeng sa phekolo ea migraine kaha, ho fapana le triptans, bahanyetsi ba CGRP ba molomo ha ba bone thepa ea vasoconstrictive 'me ka hona ba bolokehile hore ba sebelisoe ho bakuli ba nang le li-contraindications ho phekolo e tloaelehileng.
Rimegepant keCalcitoninMohanyetsi oa Mohanyetsi oa Peptide ea amanang le Gene. Mokhoa oa ts'ebetso oa rimegepant o joalo kaCalcitoninMohanyetsi oa Mohanyetsi oa Peptide ea amanang le Gene.
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